Page 65 - 76_02
P. 65

VOL. 76 (2), 259-305, 2010  UTILIZACIÓN DE HIDROLASAS EN LA PREPARACIÓN...

70. Mischitz, M., et al. (1995) Asymmetric microbial hydrolysís of epoxides. Tetra-
       hedron Asymmetry. 6: 1261.

71. Catt, J. D., et al. (1999) Preparation of benzofuran and dihydrobenzofuran
       melatonergic agents. US.5856529, CAN 130:11015.

72. Goswami, A., et al. (1999) Stercospecific enzymatic hydrolysis of racemic
       epoxide: a process for making chiral epoxide. Tetrahedron Asymmetry. 10: 3167.

73. Arch, J. R. S. (1997) $-3-adrenoceptors and other putative atypical $-adreno-
       ceptors. Pharmacol. Rev. Commun. 9: 141.

74. Bloom, J. D., et al. (1989) Disodium (R.,R) 5-[2-(3-chlorophenyl)-2-hydroxye-
       thyl] amino] propyl]-1,3- benzodioxole-2.2-dicarboxylate: a potent $-adrener-
       gic agonist virtualIy specific for $-3-receptors. J. Med. Chem. 35: 3081.

75. Fisher, L. G., et al. (1994) BMS-187257, a potent, selective, and novel hetero-
       cyclic $-3 adrenergic receptor agonist. Bioorg. Med. Chem. Lett. 6: 2253.

76. Patel, R. N., et al. (1998) Microbial synthesis of chiral intermediates for $-3-
       receptor agonists. J. Am. Oil Chem. Soc. 75: 1473.

77. Campos, F., et al. (2000) An efficient enantioselective synthesis of (R,R)-for
       formoterol, a potent bronchodilator, using lipases. Tetrahedron. Asymmetry.
       11: 2705.

78. Bisacchi, G. (1999) Preparation of amidino and guanidino azetildinone com-
       pounds as tryptase inhibitors. WO 9967215, Al 19991229, CAN 132:64103, AN
       1999:819347.

79. Wirz, B. & Walther, W. (1992) Enzymic preparation of chiral 3-(hydroxyme-
       thyl)piperidine derivatives. Tetrahedron Asymmetry. 3: 1049.

80. Goswami, A., et al. (2001) Chemical and enzymatic resolution of (R.S)-N.(tert-
       butoxycarbonyl-3-hydroxymethylpiperidine. Organic Process. R&D. 5: 415.

81. Schenk, D., et al. (2001) Potential treatment opportunities for Alzheirner’s
       disease through inhibition of secretases and A$ immunization. J. Mol. Neuros-
       ci. 17: 259.

82. Audia, J., et al. Preparation of N- (phenylacetyl)di-and tripeptíde derivatives
       for inhibiting $-amyloid peptide release. PCT lnt. Appl., WO 9822494, A2
       19980528, CAN 129:41414, 126.

83. Patel, R. N., et al. (2000) Enzymatic resolution of racemic secondary alcohols
       by lipase B from Candida antarctica. J. Am. Oil. Chem. Soc. 77: 1015.

84. Nanduri, V. B., et al. (2001) Biochemical approaches to the synthesis of ethyl
       5-(S)-hydroxyl hexanoate and 5-(S) hydroxyhexanenitrile. Enzyme Microb.
       Technol. 28 (7&8): 632.

85. Kagechika, H., et al. (1988) Retinobenzoic acids, 1: structure-activity relatio-
       nship of aromatic amides with retinoidal activity. J. Med. Chem. 31: 2182.

86. Shudo, K. & Kagechika, H. (1989) Structure-activity relationships of a new
       series of synthetic retinoids, in Chemistry and Biology of Synthetic Retinoids.
       Dawson, M. I. & Okarnura, W. H., Eds. CRC Press, Boca Raton, FL.

87. Moon, R. C. & Itri, L. M. (1984) Retinoids and cancer. Retinoids. 2: 327.
88. Kagechika, H., et al. (1988) Retinobenzoic acids, 1: structure-activity relatio-

       nships of aromatic amides with retinoidal activity. J. Med. Chem. 31: 2182.
89. Belema, M.; Zusi, F. C. & Tramposch, K. M. (2000) Active enantiomer of RAR

       ‘(-specific agonist, PCI Int. Appl. WO 0016769 Al 20000330 CAN 132:246379
       AN 2000:209902.

                            303
   60   61   62   63   64   65   66   67   68   69   70